Lactacystin, 1 mg
Product#: FNK-BLK-0460-1mg
$285.03
Availability:
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Lactacystin
Cat No:
FNK-BLK-0460-1mg
Product ID and Size
| Cat No. | Description | Size | Link |
| FNK-BLK-0460-100ug | Lactacystin | 100μg |  |
| FNK-BLK-0460-500ug | Lactacystin | 500μg | |
| FNK-BLK-0460-1mg | Lactacystin | 1mg | |
| FNK-BLK-0460-5mg | Lactacystin | 5mg | |
Description
Biological activity: 1) Lactacystin inhibits cell cycle progression and induces neurite outgrowth in Neuro 2a cells. 2) Inhibits proteasome activity. Proteasome exhibits three protease activities of the tree, Lactacystin inhibits chymotrypsin-like activity most potently, followed by trypsin-like activity, but its inhibitory activity against peptidylglutamylpeptide hydrolytic activity is relatively weak.
Origin: Streptomyces lactacystinnaeus OM-6519
CAS Registry Number: 133343-34-7
Appearance: White powder
Molecular Formula/ Weight: C15H24N2O7S=376.13
Purity: >98.0% by HPLC
Solubility: Sol. in DMSO, MeOH, EtOH, water
Handling and Storage: Store at -20℃.
References:
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- T. Sunazuka, et al., Tetrahedron Lett., 34 4447 (1993).
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